Glutamate Induced Calcium Signals in Proliferating Cells of the Central Nervous System in Adult Zebrafish Philip Merksamer Advisor: Stuart Thompson June 2003 Permission is granted to Stanford University to use the citation and abstract of this paper. Abstract The periventricular zone (PVZ) of the adult zebrafish central nervous system contains undifferentiated, proliferating cells consistent with the properties of neural progenitors. Past studies suggest that axonal projections may extend from the optic tectal neurons into the PVZ allowing for the possibility that the optic tectal neurons signal the PVZ with neurotransmitters, In this study, time-lapse confocal imaging of PVZ cells labeled with fluo-4 AM calcium indicator is employed to demonstrate that PVZ cells respond to glutamate through elevated intracellular calcium levels. The NMDA receptor antagonist, APV, and the AMPA receptor antagonist, CNQX, block this response. PVZ cells appear to express functional AMPA and NMDA receptors, and these receptors may play an important role in proliferation, migration, or differentiation of the PVZ cells. Introduction Neural progenitors are immortal cell lines capable of differentiating into mature neural tissue. Considerable amounts of research are devoted to the study of neural progenitor cells in order to elucidate the mechanism of neural regeneration as well as to develop treatments for neural degenerative disorders. Zebrafish (Danio Rario) are advantageous model organisms for such research because they generate new neurons throughout their adult lives and thus are presumed to posses neural progenitors (Thompson, unpublished data). Past studies indicate that the round cells of the periventricular zone (PVZ) in the optic tectum of adult zebrafish may be such progenitor cells. These cells have been shown to proliferate both in-vivo and in culture (Tulloch, 2002; Webster, 2002). While the morphology of the PVZ cells has been well characterized, little is known about signaling and activation of these cells. There are indications that axonal projections extend from the optic tectum into the PVZ permitting the possibility that optic tectum neurons interact synaptically with the PVZ cells (Arakaki, unpublished data). Synaptic interaction between neurons is crucial for proper CNS function. It is unknown, however, whether synaptic interaction between neurons and neural progenitors exists, and whether such interaction is necessary for neural progenitor activation and differentiation. This study addresses the question; do PVZ cells respond to the neurotransmitter, glutamate, through NMDA- and AMPA-type glutamate receptors? Glutamate signaling acting on both NMDA receptors (NMDA-R) and AMPA receptors (AMPA-R) has been shown necessary for proper development of dendritic arbors in Xenopus optic tectal neurons (Rajan & Cline, 1998). A similar mechanism may operate in the signaling of PVZ cells in zebrafish. In this study, time-lapse confocal images were taken of living optic tectum slices during the application of glutamate and glutamate receptor antagonists. These images were analyzed for increased intracellular calcium concentration using the fluorescent indicator, fluo-4 AM. An elevated intracellular calcium concentration is indicative of a response to glutamate because both AMPA-R and NMDA-R generate a rise in intracellular calcium. I find that the PVZ cells respond to glutamate through elevated intracellular calcium levels. This response is blocked by the selective NMDA-R antagonist, APV, and by the selective AMPA-R antagonist, CNOX. Methods Brain Slice Preparation. Adult zebrafish brains were dissected in Hanks media containing (mM): Nacl 96, KCI 3.78, NazHPO4 0.175, KH2PO4 0.308, CaClz 0.91, MgSO4 0.7, NaHCO; 4.2, CeHj2O6 25. The optic tectum lobes were cut from the brain and incubated with SuM of the calcium sensitive indicator, fluo-4 AM (Molecular Probes) for forty minutes, followed by a ten minute wash with either Hanks or Hanks plus the glutamate receptor antagonists APV (100 uM) or CNQX (100 uM). Confocal Microscopy. Time-lapse confocal images were taken of optic tectum slices using an Olympus microscope with a 40x water-immersion objective. Äfter the first ten frames, 1 ml of Hanks, followed by 1 ml of 10 uM glutamate, or 1 ml of Hanks, followed by 1 ml of 10 uM ionomcyin was added to the profusion dish containing the optic tectum slice. lonomycin is a calcium sensitive ionophore and was used to determine the saturation point for the fluo-4 AM indicator. Images were taken for a total of 120 frames, with approximately two seconds between each frame. Fluorescence analysis. Äfter imaging, six to ten regions of interest were sampled for fluorescence intensity vs. time. Baseline fluorescence, Fo, was defined as the average fluorescence over the first 10 frames. Fluorescence was averaged over 5 pixels and converted to units of AF/Fo. Fluorescence intensities were converted to calcium concentration (nM) from the following equation: Ca2 - Ka' (F - Fmin)/(Fmax - F) Kq, the dissociation constant for fluo-4 AM, was 345 nM. Fmax was given by the response to ionomcyin and was set to 1.6. Fmin was set to 0.826 so that an F value of 1 gives a calcium concentration of 100 nM. Results The optic tectum slices were fully saturated with fluo-4 AM indicator after incubation for one hour (Fig. 1), however, a forty minute incubation was sufficient for confocal imaging. The indicator stained only the edge of the tectum and the periventricular zone closet to the edge. The addition of the calcium specific ionophore, ionomycin, resulted in an elevated fluorescence intensity from 1 to 1.4 AF/F (Fig 2). The intracellular calcium concentration increased from a resting concentration of 104 nM to 1058 nM. The addition of glutamate resulted in elevated fluorescence intensity compared to a saline control reaching a maximum intensity of approximately 1.27 AF/F (Fig 3). The intracellular calcium concentration increased from a resting concentration of 102 nM +- 38 (95% confidence interval) to 366 +- 149 nM averaged over 16 individual cells from two independent experiments. When the optic tectum slice was incubated with the NMDA-R antagonist, APV, the addition of glutamate resulted in no elevated fluorescence intensity compared to a saline control (Fig 4). The calcium concentration increased from 100 +- 37 nM to 112 +- 38 nM averaged over eight cells. When the optic tectum slice was incubated with the AMPA-R antagonist, CNQX, the addition of glutamate resulted in a slight elevated fluorescence intensity compared to a saline control reaching a maximum intensity of 1.12 AF/F (Fig 5). Calcium concentration increased from 100 +/- 44 nM to 160 +- 76 nM averaged over 18 cells from two independent experiments. Discussion In this study, I have provided evidence that the neural progenitors of the PVZ express functional ionotropic glutamate receptors. First, I demonstrated that the PVZ cells respond to glutamate through a 3-fold increase in intracellular calcium. Second, I found that the selective antagonists, APV and CNQX blocked this elevated calcium response. Because APV and CNOX specifically block NMDA-R and AMPA-R respectively, the cells in the PVZ contain both types of receptors. There is considerable evidence that embryonic mammalian cells within ventricular zones (VZ) express many amino acid neurotransmitters and their respective receptors (Lo Turco et al., 1991 & 1995). However, not all mammalian VZ cells proliferate, and some precursor cells begin differentiation in the ventricular zone (Li et. al., 1998). Furthermore, using a calcium imaging technique similar to this study, Maric et. al. found evidence that AMPA/kainate receptors first appear in the terminal cell division stage of embryonic neural precursor cells and may be involved in differentiation and commitment to a neuronal cell lineage (2000). In this study, there was considerable variability in the glutamate response of PVZ cells (366 + 149). This variability could have a physiological basis in that not all the cells of the PVZ may express ionotropic glutamate receptors. It is possible that only a subset of PVZ cells that have begun to differentiate are expressing such receptors which would be consistent with previous findings in mammalian systems. It is also possible, however, that the variability was due to the experimental design. The quality of staining with fluo-4 AM was not consistent, and sometimes the PVZ cells would not take up the indicator. This study could be bolstered with more experiments, particularly one using the agonists, AMPA and NMDA. An elevated calcium response to AMPA and NMDA would provide strong supporting evidence that the PVZ cells express functional AMPA and NMDA receptors. Also, an in-situ hybridization analysis for mRNA transcripts encoding AMPA and NMDA submit genes would furnish further evidence that these receptors are actively expressed. Finally, the extent to which the ionotropic glutamate receptors are involved in proliferation, migration, and differentiation in the PVZ cells remain unknown. However, the existence of such receptors and the fact that they cause elevated cytosolic calcium levels implies that glutamate acting on ionotropic receptors has a considerable role in PVZ cell signaling. Conclusion Using time-lapse confocal imaging, this study demonstrated that the PVZ cells considered to be neural progenitors respond to glutamate through elevated calcium levels. The antagonists, APV and CNQX, blocked this response, indicating that the PVZ cells express functional NMDA- and AMPA-receptors. The ionotropic glutamate receptors thus appear to be involved in cell signaling in the PVZ, however it is still unknown whether these receptors are directly involved in proliferation, migration, or differentiation, three critical features of progenitor cells. Literature Cited Li W, Cogswell CA, Lo Turco JJ. 1998. Neuronal differentiation of precursors in the neocortical ventricular zone is triggered by BMP. J Neurosci 18:8853-8862. Lo Turco JJ, Blanton MG, Kriegstein AR. 1991. Initial expression and endogenous activation of NMDA channels in early neocortical development. J Neurosci 11: 792-799. Lo Turco JJ, Owens DF, Heath MJS, Davis MBE, Kriegstein AR. 1995. GABA and glutamate depolarize cortical progenitor cells and inhibit DNA synthesis. Neuron 15:1287-1298. Maric D, Liu QY, Grant GM, Andreadis JD, Hu Q, Chang YH, Barker JL, Joseph J, Stenger DA, Ma W. 2000. Functional ionotropic glutamate receptors emerge during terminal cell division and early neuronal differentiation of rat neuroepithelial cells. J Neurosci Res. 61:652-62. Rajan I, Cline HT. 1998. Glutamate receptor activity is required for normal development of tectal cell dendrites in vivo. J Neurosci 18:7836-7846 Tulloch, N. 2002. In vitro growth of zebrafish neural precursors. Unpublished MS on file at Hopkins Marine Station Library. Webster, B. 2002. Insulin-like growth factor I and fibroblast growth factor modulate neural progenitor cell proliferation in the adult zebrafish brain. Unpublished MS on file at Hopkins Marine Station Library. Appendix 1 All References Cameron HA, Hazel TG, Mckay DG. 1998. Regulation of neurogenesis by growth factors and neurotrasnmitters. J Neurobiol 36:287-306. Ciccolini F, Collins TJ, Sudhoelter J, Lipp P, Berridge MJ, Bootman MD. 2003. Local and global spontaneous calcium events regulate neurite outgrowth and onset of GABAergic phenotype during neural precursor differentiation. J Neurosci. 23:103-11. Gleason EL, Spitzer NC. 1998. AMPA and NMDA receptors expressed by differentiating Xenopus spinal neurons. J Neurophysiol 79:2986-2998. Komuro YH, Rakic P. 1993. Modulation of neuronal migration by NMDA receptors. Science 260:95-97. Li W, Cogswell CA, Lo Turco JJ. 1998. Neuronal differentiation of precursors in the neocortical ventricular zone is triggered by BMP. J Neurosci 18:8853-8862. Lo Turco JJ, Blanton MG, Kriegstein AR. 1991. Initial expression and endogenous activation of NMDA channels in early neocortical development. J Neurosci 11: 792-799. Lo Turco JJ, Owens DF, Heath MJS, Davis MBE, Kriegstein AR. 1995. GABA and glutamate depolarize cortical progenitor cells and inhibit DNA synthesis. Neuron 15:1287-1298. Maric D, Liu QY, Grant GM, Andreadis JD, Hu Q, Chang YH, Barker JL, Joseph J, Stenger DA, Ma W. 2000. Functional ionotropic glutamate receptors emerge during terminal cell division and early neuronal differentiation of rat neuroepithelial cells. J Neurosci Res. 61:652-62. Mitsui K, Tokuzawa Y, Itoh H, Kohichi S, Murakami M, Takahashi K, Maruyama M, Maeda M, Yamanaka S. 2003. The homeoprotein nanog is required for maintenance of pluirpotency in mouse epiblast and ES cells. Cell 133:631-642. Rajan I, Witte Sm Cline HT 1999. NMDA receptor activity stabilizes presynaptic retinotectal axons and postsynaptic optic tectal cell dendrites in vivo. J Neurobiol 38:357-368 Rajan I, Cline HT. 1998. Glutamate receptor activity is required for normal development of tectal cell dendrites in vivo. J Neurosci 18:7836-7846 Tulloch, N. 2002. In vitro growth of zebrafish neural precursors. Unpublished MS on file at Hopkins Marine Station Library. Webster, B. 2002. Insulin-like growth factor I and fibroblast growth factor modulate neural progenitor cell proliferation in the adult zebrafish brain. Unpublished MS on file at Hopkins Marine Station Library. Wu G-Y, Malinow R, Cline HT 1996. Maturation of a central glutamatergic synapse. Science 274:972-976. Wullimann M, Rupp B, Reichert H. 1996. Neuroanatomy of the Zebrafish Brain. Birkhauser Verlag, Basel, Switzerland. Appendix 2: Figures Normalized Average Intensity vs. Time After Dye Loading 10 Time (10 Minute Intervals) Figure 1: Average intensity vs. Time after dye loading. AF/Fvs. Time 1.6 1.4 — Control 1 lonomycin 1OuM 0.9 0.8 150 200 100 50 time (sec) Figure 2: AF/F vs. Time for the Negative Control (saline) and the positive control (ionomycin). Calcium Response to Glutamate — Contro Glutamate10UM 0.9 0.8 - 50 100 150 200 250 300 time (sec) Figure 3: AF/F vs. Time for the negative control and glutamate. Calcium Response to Glutamate in the presence of APV (T00uM) 1.6 1.4 + 1.3 — Contro Glutamate 10UM 0.9 0.8 - 50 100 150 200 250 300 time (sec.) Figure 4: AF/F vs. Time for control and glutamate in the presence of APV. Calcium Response to Glutamate in the Presence of CNOX (100uM) — Control Glutamate 10uM lonomycin 10uM 0.9 0.8 0 50 100 150 200 250 300 time (seo Figure 5: AF/F vs. Time for control, glutamate, and ionomycin in the presence of CNOX. 600 500 400 Conto Glutamate 300 □ Glutamate with APV EGlutamate with CNOX 100 Figure 6: Bar Graph comparing calcium concentration for each treatment.