Erica Li Bio 175H: Problems in Ecology and Ecophysiology Advisor: Epel Bisphenol A causes disruptions in the cell cycle of the zygotes and embryos of the purple sea urchin, Strongylocentrotus purpuratus Abstract Bisphenol A (BPA), a common chemical found in polycarbonate plastic containers, is suspected to damage animal health. While many studies on BPA have been done on terrestrial vertebrate models, few have been conducted on marine invertebrates Because BPA is found in harbours, it is important to find out if we need to be concerned about BPA pollution of the marine ecosystem. This study examines the effects of BPA on the early development of the purple sea urchin, Strongylocentrotus purpuratus. The results show that the vast majority of the embryos develop normally when exposed to concentrations at or below 1 uM up to the late prism stage; a few exogastrulating embryos appear as a result of BPA exposure, but the number of exogastrulating embryos does not increase with increasing concentration. BPA inhibits formation of the blastocoel in S. purpuratus embryos at concentrations greater than 1 uM. At concentrations greater than 5 uM, BPA significantly delays cell division, apparently affecting the mitotic apparatus of the zygote and preventing chromosomes from condensing and migrating properly. The concentrations used in this study are orders of magnitude higher than what has been found in the environment, indicating that BPA may not be of concern in marine ecosystems. Erica Li Bio 175H: Problems in Ecology and Ecophysiology Advisor: Epel Bisphenol A causes disruptions in the cell cycle of the zygotes and embryos of the purple sea urchin, Strongylocentrotus purpuratus Abstract Bisphenol A (BPA), a common chemical found in polycarbonate plastic containers, is suspected to damage animal health. While many studies on BPA have been done on terrestrial vertebrate models, few have been conducted on marine invertebrates. Because BPA is found in harbours, it is important to find out if we need to be concerned about BPA pollution of the marine ecosystem. This study examines the effects of BPA on the early development of the purple sea urchin, Strongylocentrotus purpuratus. The results show that the vast majority of the embryos develop normally when exposed to concentrations at or below 1 uM up to the late prism stage; a few exogastrulating embryos appear as a result of BPA exposure, but the number of exogastrulating embryos does not increase with increasing concentration. BPA inhibits formation of the blastocoel in S. purpuratus embryos at concentrations greater than 1 uM. At concentrations greater than 5 uM, BPA significantly delays cell division, apparently affecting the mitotic apparatus of the zygote and preventing chromosomes from condensing and migrating properly. The concentrations used in this study are orders of magnitude higher than what has been found in the environment, indicating that BPA may not be of concern in marine ecosystems. Introduction Bisphenol A (BPA) is gaining attention for its ability to interfere with the health of animals. It is a common industrial chemical, found in polycarbonate plastics that are used for lab flasks, animal cages, and many consumer products such as drinking water jugs and bottles. (Colborn et al, 1996) As a xenoestrogen, BPA is many orders of magnitude less potent than estradiol. (Milligan et al, 1998) However, according to David Feldman, a professor of medicine in the endocrinology division of the Stanford School of Medicine, it "still has activity in the parts per billion range." (Colborn et al, 1996) BPA is also present in relatively high concentrations- as high as eighty parts per billion—in canned foods, such as canned corn, artichokes, and peas. (Colborn et al, 1996) A number of studies have been done on terrestrial vertebrate model organisms to ascertain the health-damaging effects of BPA, some with seemingly conflicting results. Masaru Furuya et al showed that dietary BPA at 200 mg per rooster per week feminizes roosters. (Furuya et al, 2003) According to a multi-generation study conducted by Rochelle Tyl et al, dietary BPA did not significantly damage the health of Sprague-Dawley rats or the health of their offsprings. (Tyl et al, 2002) A study on mice by Patricia Hunt et al, however, demonstrated that BPA causes meiotic aneuploidy in the oocytes of female mouse. (Hunt et al, 2003) Possibly related to this, Lehmann and Metzler concluded that Bisphenol A interferes with microtubules in cultured human fibroblasts. (Lehmann and Metzler, 2003) In a study on a variety of chemicals suspected to cause aneuploidy, Parry et al demonstrated that bisphenol A induces aneuploidy in Chinese hamster V79 cells at 14 ug/ml. There was a dose-dependent increase in the frequencies of both abnormal metaphases and all mitotic aberrations when those cells were exposed to BPA. Parry et al concluded that BPA may interact with components of the centrosomes which make up the poles of the mitotic spindle. (Parry et al, 2002) Less attention has been paid to how BPA affects organisms in aquatic systems. In one study by H. Segner et al on the freshwater zebrafish, Danio rerio, BPA was shown not to be a potent xenoestrogen. (Segner et al, 2003) However, no BPA study has been conducted on marine invertebrate model organisms, despite the fact that a nationwide investigation of endocrine disruptors in Japan’s harbors, conducted by Hosokawa et al, found BPA in at least thirty percent of the sites surveyed. (Hosokawa et al, 2003) It is thus relevant to examine the effects of bisphenol A on a marine invertebrate model organism in order to ascertain whether the scientific community and policy makers need to be concerned about BPA pollution of marine systems. The studies by Hunt, Lehmann and Metzler, and Parry suggest that it is worthwhile to examine the effects of BPA on cell division. The experiments described below were designed to examine how BPA affects cell division and differentiation in the early development of the sea urchin, Strongylocentrotus purpuratus. The results show that BPA at concentrations above 5 uM disrupts S. purpuratus development by affecting mitosis even at the fertilized one-cell stage. Embryos exposed at 3 uM of BPA divide slower than the controls and never form the blastocoel, possibly due to disruptions of the mitotic apparatus. In contrast, embryos exposed to 1 uM of BPA or less develop normally till at least the late prism stage. Materials and Methods General protocols common to all three parts of the experiment A O.1M stock solution of bisphenol A was made in DMSO, stored at room temperature in a covered graduated cylinder, and shielded from light with tin foil. All dilutions of the stock solution were done using filtered seawater. Sea urchins (Strongylocentrotus purpuratus) were induced to spawn by injection with approximately 1 mL of O.5M potassium chloride into the coelomic cavity. Females were placed upside-down on top of a small beaker (beaker diameter smaller than the diameter of the urchin) filled with sea water, such that eggs fell to the bottom of the beaker. The eggs were stored in the cold room at 16 °C and could be used for about two days. Sperm was pipetted from the dorsal side of the males directly into an eppendorf tube and stored in the refrigerator at 4 °C. The density of zygotes in the culture was low such that the zygotes would not get anoxic To achieve this, about 0.2 mL of super-concentrated egg suspension was diluted in a beaker containing 500 mL of filtered sea water. Fifteen minutes after 5 uL of sperm was added to the eggs in BPA-free sea water, the eggs were checked under the microscope to see if they possessed the fertilization envelope. If more than 90% of the eggs were fertilized, they were exposed to control and experimental conditions, described below. Part one: does BPA affect the developmental schedule of S. purpuratus embryos up to the late prism stage? Fertilized zygotes were placed in covered glass petri dishes containing 10 mL of sea water and various concentrations of BPA ranging from O.1 uM to 1 mM. The control group was kept in the same kind of petric dishes with the same volume of sea water, but without any BPA. Sperm from three males were used to fertilize the eggs of one female. Thus, for each concentration of BPA, there were three samples total. The zygotes were checked by light microscopy at 15 minutes, 2 hours, 4 hours, 6 hours, 20 hours, 23 hours, 46 hours, 49 hours, and 70 hours after fertilization. In between sampling, the embryo cultures were left in a cold room maintained at 16 °C. When this part of the experiment was repeated, fertilized zygotes were placed in glass test tubes that were covered with parafilm. The test tubes rested on a rack in the 16 C cold room. Part two: does BPA affect the cell division schedule The experiment was conducted in glass test tubes containing control, 1 uM, 3 uM, 5 uM, and 7 uM of BPA. The other conditions were the same as those described in Part One. Pure DMSO was diluted 100 times with filtered seawater and added to the control group, such that the control group had the same amount of diluted DMSO as the sample with the highest amount of BPA. Fertilized embryos were added to each test tube and checked using light microscopy about every 30 minutes until the control group arrived at the morula stage. Part three: BPA’s effect on chromosome appearance during the first cleavage A solution containing 7 uM of BPA was made. Eight Falcon polystyrene test tubes were filled with 10 mL of control samples each. Another eight tubes were filled with embryos exposed to 7uM of BPA. The 16 tubes were placed on a rocker table for 1 hour at room temperature. Then, every 15 minutes, one control and one experimental sample were taken and centrifuged in a hand-crank low-speed centrifuge such that the embryos settled at the bottom of the test tubes. The liquids from the two tubes were aspirated. 5 mLs of Carnoys solution (1 part glacial acetic acid: 3parts ethanol) was added to both tubes, and the samples were placed on a test tube rack at room temperature. This process was repeated until all eight sets of zygotes were fixed in Carnoys. After approximately 24 hours, the Carnoys solution was aspirated from all test tubes. All zygotes were placed in 45% acetic acid for about 30 minutes. The acetic acid was then removed and a solution of 2% acetocarmine with 45% acetic acid was added to all samples. After 10 minutes, the cell samples were placed on a slide under a phase microscope and examined for chromosome arrangement. Results Part one: does BPA affect the life stage schedule of S. purpuratus embryos up to the late prism stage! A vast majority of S. purpuratus embryos were able to grow to at least the late prism stage in BPA concentrations less than or equal to 1 uM. At concentrations greater than 3 uM, however, 100 % of the embryos failed to develop a blastocoel and to make it past the morula stage. At concentrations above 25 uM, embryos lysed and died early at the 1-cell stage. Concentrations of 3 uM, 6 uM, and 10 uM caused development to be delayed. Problems with cell division were seen in the 3 uM group at 2 hours after fertilization, when the zygotes were going through the first cleavage. Many of the zygotes exposed to 3 uM had various problems such as asynchronous cell division, wrong number of cells, and incomplete cytokinesis. The developmental progress of the 6 uM, and 10 uM groups was delayed further than the 3 uM group, and the morphological abnormalities were more prominent. At 2 hours after fertilization, there were some normal-looking zygotes at the 2-cell stage in the 3 uM group, but none in the groups exposed to 6 uM of BPA or more. Even though embryos exposed to 3 uM, 6 uM, and 10 uM of BPA displayed delays and abnormalities at 2 hours after fertilization, their cells continued to divide abnormally and many survived till at least the third day after fertilization. At 76 hours, some embryos exposed to 10 UM of BPA were swimming, even though they were dumbbell shaped and completely abnormal There were no exogastrulates in the control groups. In all experimental groups up to 1 UM, there were a few exogastrulating individuals. The number of exogastrulates and the degree of exogastrulation did not seem to vary significantly with varying concentrations. Part two: does BPA affect the cell division schedule Given the above observation that BPA concentrations at greater than 3 uM delay development, a study was conducted to see if BPA delays cell-division. It was observed that at about 2 hours after fertilization, the control, 1 uM, and 3 uM groups were all predominantly at the 2-cell stage. The cell division schedule in the 5 uM group was delayed—one could see the cells in the process of dividing but cytokinesis had not yet happened at 2 hours. In the 7 uM group at this time, all zygotes were completely at the 1-cell stage, looking round. At about 2.5 hours after fertilization, the control and 1 uM groups looked mostly healthy. Both groups had approximately equal numbers of 2-cell and 4-cell stage embryos. Cell division abnormalities started emerging in the 3 uM group at this time, though many of the embryos also made it to normal 2-cell and 4-cell stages. The 5 uM group was clearly developmentally behind the groups with lower concentrations. Most of the embryos exposed to 5 uM BPA were still at the 1-cell or 2-cell stages, and the ones that were beyond the 2-cell stage clearly had incomplete cytokinesis and unequal divisions. (Fig. 1) In the 7 uM group, there were hardly any discernible boundaries between cells. Most of the zygotes could be categorized as being at the 1-cell stage, but there were invaginations in the cell membrane and the zygotes were no longer round. Each embryo in this group contained fewer cells than the embryos of the other groups. At about 3.5 hours after fertilization, the control group was predominantly at the 8-cell stage. The 3 uM and 5 uM groups had predominantly abnormal zygotes with 8 or more cells. The 7 uM group, in contrast, had mostly morphologically abnormal zygotes that clearly had less than 8 cells. At about 4 hours after fertilization, the control, 1 uM, and 3 uM groups were apparently at the morula stage, whereas the 5 uM group contained comparatively less cells and more deformities. The 7 uM group was delayed even further. It had more cases of incomplete cytokinesis and more morphologically deformed cells than the 5 uM group. Later on, all the zygotes looked like they were at the morula stage and it became impossible to visually discern how many cells an embryo had. The sheer number of cells also made it impossible to clearly discern the morphology of the cells, and all the samples started appearing similar to one another. At this point, the experiment was halted. Part three: how does BPA affect cell division In this third study, I examined in more detail the inhibition of cell division. At first the control and experimental group appeared similar. (Fig. 2 and 3) At about 1.75 and 2 hours after fertilization, the chromosomes in some of the zygotes in the control group began to organize in two sets, lined up, and migrated to one side of the zygote. The chromosomes of all zygotes in the experimental group still appeared scattered and more near the center of the zygote. (Fig. 4) At 2.25 and 2.5 hours after fertilization, some of the zygotes in the control group showed clear division and arrived at the 2-cell stage, whereas no 2-cell stage zygotes could be found in the experimental group. In the control group, two sets of chromosomes could be seen in some zygotes, but in all experimental zygotes only one set of chromosomes could be seen. (Fig. 5 and The result from this part of the experiment was problematic in that not all zygotes in the control group divided. In the samples where the zygotes did divide, the cleavage furrow was often difficult to discern, making visualizing two sets of chromosomes the only indication of cell division. Oftentimes, only one set of chromosome was found in the zygotes of the control group, which was possibly confounded by the fact that the fixing and staining technique described did not yield extremely clear images of the chromosomes. Nonetheless, there was a difference in chromosome morphology between the control and experimental groups. It was significant that no zygote in the experimental group divided in 2.5 hours, whereas at least some divided in the control group. Discussion The experiments demonstrate that S. purpuratus embryos are able to develop normally up to the late prism stage in BPA concentrations up to 1 uM. At concentrations equal and above 3 UM, BPA delays development, inhibits blastocoel formation, delays cell division, and affects chromosome arrangement during mitosis. However, concentrations up to 10 uM of BPA are not immediately lethal, and abnormal embryos continue to experience cell division despite the failure to form the blastocoel until at least 70 hours after fertilization. The individual exogastrulates are difficult to explain. None existed in the control group. but the number of exogastrulates did not increase significantly with increasing concentration. As the exogastrulates were greatly in the minority, it is difficult to draw conclusions regarding the effects of BPA on exogastrulation. It would be helpful to repeat each part of the experiment a few more times and perform them in a more streamlined, consistent way. Compared to past studies and publications, some of the results from this study are surprising. Hunt et al concluded that “low-dose BPA exposure... is sufficient to cause meiotic abnormalities." (Hunt et al, 2003) Hunt et al fed the mice bisphenol A at 20, 40, or 100 ngg body weight/day for 6-8 days preceding oocyte analysis. To determine the shortest exposure that produced detectable effects, another set of experiments using a dose of 20 ng BPA/g body weight for 3, 5, or 7 days prior to oocyte analysis was conducted. From these experiments, Hunt et al concluded that BPA causes aneuploidy in the oocytes of female mice even at low doses. In my experiment, I cannot feed BPA to sea urchin embryos using ng BPA/ body weight because the embryos are too small. For the purpose of our discussion, we shall use the weight of the sea water surrounding the embryos in the denominator and assume that an embryo's body is also predominantly water. The molecular weight of BPA is 228.29. Calculations show that if Hunt et al fed BPA to mice at 20 ng BPA/ g mice body weight, then they were feeding 8.76 x 10 moles of BPA to each kilogram of mice. Assuming the density of animal body and water are approximately the same, the concentration at which Hunt et al achieved an effect was 8.76 x 10 M. The lowest concentration where my experiment achieved a clearly discernible effect was 3 x 10° M. Thus, Hunt’s effective concentration was about 33 times lower than mine. However, because BPA is practically insoluble in water, it may accumulate in the fatty tissues of the mice. This may explain the extremely low effective concentration presented in Hunt et al’s study. Remarkably, in the study conducted by Parry et al, an effectively aneugenic concentration of BPA was as high as about 40 uM. (Parry et al, 2002) At such concentration, Parry et al showed that dividing cells became multipolar because the chemical may have interacted with components of the centrosomes that make up the poles of the mitotic spindle. In contrast to Parry et al’s finding, my experiments show that 40 uM of BPA would kill the S. purpuratus embryos instantly. In addition, according to Tyl et al, BPA damages the health of SD rats at only above 750 ppm. (Tyl et al, 2002) This concentration is equal to 3.285 x 10 M, which, like Parry's effective concentration, is significantly higher than the concentration that inhibits blastocoel formation in sea urchin embryos. The wide differences among effective concentration shown by the aforementioned studies suggest that there may be species-dependent factors regarding vulnerability to BPA. The levels of BPA that affect mice, rats, and hamsters, three species of rodents, are completely different. 11 Furthermore, concentration that affects the early development of sea urchins is different from the concentrations that affect any of the rodent species in the aforementioned studies. Because marine life is extremely diverse, one must take care when attempting to extrapolate the sea urchin embryo data to other species. The environmental relevance of the concentrations used in my sea urchin embryo study should also be discussed. In an environmental study on BPA, the brother and sister team of Fatima Olea, a food toxicologist, and Nicolas Olea, a physician specializing in endocrine cancers, found BPA in canned vegetables at 80 parts per billion. "At such levels," wrote Theo Colborn and her co-authors of Our Stolen Future, “a synthetic estrogen mimic might contribute significantly to a person’s exposure regardless of whether it is a "weak" estrogen or not.' (Colborn et al, 1996) 80 ppb of BPA was cause for human health concerns. However, assuming that canned vegetables are mostly made of water, 80 ppb of BPA translates into a concentration of 3.504 x 10 M, nearly an order of magnitude lower than the concentration that inhibited blastocoel formation in S. purpuratus embryos. While the report by Hosokawa et al did not mention the concentration of BPA that was found in harbors, it is unlikely that marine concentrations of BPA would exceed that found in manufactured foods. Thus, the fact that 3 uM of BPA inhibits blastocoel formation in sea urchin embryos may not be environmentally relevant, as marine life forms are probably not likely to encounter such high concentrations. Sea urchin embryos show considerable tolerance to 1 uM of BPA up to the prism stage, demonstrating the robustness of early embryos. However, it is unclear whether early exposure to BPA would affect later development. It would be important to conduct future experiments by using lower concentrations, by culturing the embryos to later life stages, and by using other marine model organisms. This study is one of the few that focuses on the effects of bisphenol A on aquatic organisms, and possibly the first that explores the effects of BPA on the early development of a marine invertebrate species. The findings raise questions regarding the action of BPA on different model systems, and prompt further investigation on the mechanisms and concentration ranges through which BPA affects animal and human health. Acknowledgements Thank you, Professor Epel, for your guidance, patience, resource books, inspiration, and butt-kicking. Thank you, Rebecca Vega, for all your patience when I interrupt your work, and for your suggestions and demonstrations. Thank you, Amro Hamdoun, for teaching me the lab etiquettes. Literature Cited Colborn, Theo, Dianne Dumanoski, and John Peterson Myers,1996. Bisphenol A. pp. 130-131, 135 in Our Stolen Future. Penguine Books USA. Czihak, G. 1975. The Sea Urchin Embryo: Biochemistry and Morphogenesis. Springer- Verlag Berlin Heidelberg, New York. Furuya, Masaru; Fumihiko Sasaki, Amin M.A. Hassanin, Sachi Kuwahara, Yasuhiro Tsukamoto. 2003. Effects of bisphenol-A on the growth of comb and testes of male chicken. Can J Vet Res. January 2003; 67 (1): 68-71 Hunt, Patricia, Kara E. Koehler, Martha Susiarjo, Craig A. Hodges, Arlene Ilagan, Robert C. Voigt, Sally Thomas, Brian F. Thomas, and Terry J. Hassold. 2003. Bisphenol A Exposure Causes Meiotic Aneuploidy in the Female Mouse. Current Biology, Vol. 13, 546-553. Lehmann, L.; Metzler, M. 2003. Bisphenol A interferes with microtubules in cultured human fibroblasts. Toxicological Sciences; v.72, no.S-1, p.254. Milligan, S. R., Balasubramanina, A. V., and Kalita, J.C. 1998. Relative potency of xenobiotic estrogens in an acute in vivo mammalian assay. Environmental Health Perspect. 106, 23-26 Parry, E.M.; J.M. Parry, C. Corso, A. Doherty, F. Haddad, T.F. Hermine, G. Johnson, M. Kayani, E. Quick, T. Warr and J. Williamson. November 2002. Detection and characterization of mechanisms of action of aneugenic chemicals. Mutagenesis, Vol. 17, No. 6, 509-521. Segner, H.; Navas, J.M.; Schaefers, C.; Wenzel, A. March 2003. Potencies of estrogenic compounds in in vitro screening assays and in life cycle tests with zebrafish in vivo. Ecotoxicology and Environmental Safety; v. 54, no. 3, pp. 315-322 Tyl, R.W., C. B. Myers, M.C. Marr, B.F. Thomas, A.R. Keimowitz, D.R. Brine, M.M. Veselica, P.A. Fail, T.Y. Chang, J.C. Seely, R.L» Joiner, J.H. Butala, S.S. Dimond, S.Z. Cagen, R.N. Shiotsuka, G.D. Stropp, and J.M Waechter. 2002. Three-Generation Reproductive Toxicity Study of Dietary Bisphenol A in CD Sprague-Dawley Rats. Toxicological Sciences 68, pp. 121-146. Yokota, Yukio.; Valeria Matranga; Zuzana Smolenicka. 2000. p. 84, pp. 206-207 in The Sea Urchin: From Basic Biology to Aquaculture. A.A. Balkema Publishers. aaa- 8. . . kaiaaa 2 Figure legends Fig. 1 Some anomalies caused by xenobiotics during the first cleavage: A: normal cleavage; B: slightly asynchronous cell cycles of the 2 blastomeres; C 2 unequal blastomeres, incomplete cleavage; D: three blastomeres, of different sizes. (Y. Yokota et al, 2000. p. 84) Many of the embryos in experimental groups with BPA concentration equal to or greater than 3uM have morphologies resembling B-D at the 2-cell stage. Effects most prominent in groups with concentration greater than 5 uM. Fig. 2. Control and experimental zygotes fixed in Carnoys and stained with acetocarmine at 35 minutes after fertilization. The experimental group is exposed to 7uM of BPA Note the similarities between the two zygotes, and the fact that chromosomes were not readily visible. Fig. 3. Control and experimental zygotes fixed in Carnoys and stained with acetocarmine at 1.25 hours after fertilization. Not much difference can be discerned between the two groups. Chromosomes scattered near the middle of the zygote in both groups. Fig 4. Control and experimental zygotes 2 hours after fertilization. Note the lining up of the chromosomes in the control group, and the scattering of the chromosomes in the experimental sample. Fig 5. Control and experimental zygotes 2.25 hours after fertilization. Note the cleavage furrow in the control group. The control group also has two sets of chromosomes. The chromosomes in the experimental sample is still scattered. Fig 6. Control and experimental zygotes 2.5 hours after fertilization. The control sample pictured is almost ready to enter the 4-cell stage—the two sets of chromosomes are lined up to divide again. The experimental, in contrast, dwells in the 1-cell stage. Its chromosomes are still scattered and not lined up, showing that the cell is still at prophase. Fig. 1 Fig. 2 Control Experimental Fig. 3 Control Experimental Fig. 4 Control Experimental Fig. 5 Control Experimental Fig. 6 Contro Experimental