The Pathways of Nitrogen Excretion in Littorina Planaxis Robert Moulton May 30, 1964 Hopkins Marine Station Pathways of Nitrogen Excretion in Littorina planaxis In the kidneys and livers of animals having ureotelic mechanisms of excretion, according to Clementi (1915; 1918), the enzyme arginase, important in urea formation through the Krebs ornithine cycle, is present in high concentration, whereas those which have a uricotelic mechanism have a much lower concentration of this enzyme and possess other enzymes such as xanthine oxidase which is important in the formation of uric acid from purines synthesized from amino acids. These organisms may also possess the additional enzymes dricase and urease to degrade the uric acid which is formed from the purine bases to urea and ammonia (Needham and Baldwin 1934). This study will show that Littorina planaxis falls into the category of uricotelic organisms since much of this organism's waste nitrogen is first converted to uric acid. Estimations of specific enzymes such as xanthine oxidase can give some insight into the possible excretory pathways involved. In addition, since many organisms continue the degradation of uric acid into simpler compounds before excretion, tests for uricase and urease are of importance so that a clear understanding of the overall excretory process may be obtained. Experimental Procedure The essential basis of all the methods which have been employed for the detection of arginase, uricase, urease, and xanthine oxidase consisted in following the conversion of the substrates arginine, uric acid, urea, and hypoxanthine respectively. In each test, 2- approximately 25 kidneys or digestive glands were minced in artificial sea water (McLeod, Onofrey, and Norris 1954) adjusted to pH 7.0 and then distributed among 10 test tubes in 0.5 ml aliquots. Substrate was added and the activity of any enzyme which may have been present was stopped by the addition of dilute sulfuric acid and sodium tungstate solution, the final solution having a pH of 7.0. In each test, a set of controls containing tissue extract or substrate alone were run simultaneously and treated in the same manner as described above. An arginine monohydrochloride solution, .85 M, was prepared and the pH adjusted to 7.0 by the addition of 10% NaoH solution. The urea substrate was prepared by dissolving 6 grams in 100 ml of artificial sea water to make a.1 M solution. Uric acid, 16.8 grams, was dissolved in 50 ml of artificial sea water to make a.2 M solution. This solution was prepared fresh before each series of tests. Hypoxanthine, 68 mg, was added to 10 ml of .05 M NaoH to make a .85 M hypoxanthine solution at pH 8.3. Ammonia was detected by Nesslerization (Haden 1923). Urea was detected similarily after treatment with urease (Sumner 1926). Uric acid was assayed by the method of Benedict (1924). All colorimetric measurements were made in a Klett-Summerson Photo- electric colorimeter. Arginase activity was estimated by following the production of urea from arginine. Xanthine oxidase activity was estimated by following the production of uric acid from hypoxanthine. Uricase activity was estimated by following the decrease in uric acid. Urease activity was estimated by following the production of -3 - ammonia from urea. Results and Discussion The results of the experiment are presented in Table 1. Arginase, an enzyme present in most terrestrial organisms, could not be detected in any of the tests performed on Littorina planaxis indicating that the formation of urea arises through pathways other than the Krebs ornithine cycle. To account for the relatively large amounts of urea excreted, the breakdown of uric acid seems to be an excellent possibility. It is possible that synthesis of less oxidized purine compounds such as hypoxanthine and xanthine from amino acid nitrogen could provide xanthine oxides. Xanthine oxidase would deal not only with the nitrogenous compounds ultimately derived from nucleic acid catabolism, but also with nitrogen derived from protein catabolism as well. An active xanthine oxidase was found to be present in the kidney tissue of this snail. Therefore, the majority of the uric acid produced within the snail could be accounted for through the metabolism of purine bases either ingested and degraded directly or synthesized from other nitrogenous compounds. Table 2 shows that the degradation of uric acid by way of uricase leads to the production of ammonia. This conversion indicates that allantoinase and allantoinase are present as well as the assayed urease. These snails appear to have specialized more than many invertebrate groups in the production of uric acid as a nitrogenous end product as can be seen from the results of these tests and those of Needham and Baldwins' (1934). These tests also show that further degradation of uric acid does in fact occur with the help of the enzymes uricase 27 4 - and urease which are both present and which are responsihle for the two important end products, urea and ammonia. The uricolytic cycle has been well worked out by Florkin and Ducha'teau (Florkin, 1960). The first stage in the process of uricolysis consists in the oxidation of uric acid itself to the more soluble substance, allantoin, under the influence of uricase. Allantoin is further degraded through a series of steps. The urea produced in this eycle is further degraded by the action of urease which is present in significant amounts in the snail Littorina planaxis to give ammonia. The majority of the conversions takes place within the kidney- heart complex. The digestive gland tissue failed to show significant enzymatic activity. Furthermore, the existence of these enzymes in the kidney could possibly be an evolutionary adaptation allowing the snails to produce excretory products according to the availability of water. This mechanism may also be an intermediate step toward terrestrial life. Summary 1. An account is given of the experiments designed to elucidate the sources and modes of formation of the excreted urea, uric acid, and ammonia in the marine gastropod Littorina planaxis. 2. It is suggested that arginase is not concerned with the production of urea in the members of this species because no correlation was found between the amount of urea and arginase activity. In the production of urea and ammonia, which represent the principal nitrogenous end products of the Littorines, the enzyme arginase is not of significant importance. 3. Xanthine oxidase is shown to present in the kidney of this snail, though hitherto, it has not been found in other marine invertebrates. (Baldwin and Needham 1934). It is suggested that this enzyme maybe responsible for formation of uric acid in Littorina planaxis and other members of this group, whether the uric acid is derived ultimately from nucleic acid breakdown or from protein deamination. 4. The uricotelic character of the metabolism of this gastropod is supported by the presence of urease, uricase, and xanthine oxidase in the kidney tissue and indicate a mechanism which can account for most of the nitrogen excretory products. Table 1 All values in mg of substrate converted Final Initial Incubation Enzyme time Arginase Argine control .009 .010 16 hr trial .009 .006 16 hr trial 2 Arginine-kidney 008 16 hr .014 trial ! .018 .010 16 hr trial 2 Kidney control .010 .010 16 hr trial .009 .013 16 hr trial 2 Arginine control .009 .008 16 hr trial ! .008 .007 16 hr trial Arginine-Dig. Gland .015 16 hr trial ! .012 .014 16 hr trial 2 .012 Dig. Gland control .011 16 hr .010 trial .008 16 hr .012 trial Xanthine oxidase Hypoxanthine control 0005 8 hr .0003 trial .000 0006 8 hr trial Hypoxanthine-kidney .0005 .0013 8 hr trial .0013 .0003 8 hr trial2 Kidney control .0002 trial 0001 8 hr .0001 8 hr .0002 trial Hypoxanthine control .0005 16 hr .0007 trial! 0008 trial 2 16 hr .0007 ypoxanthine- Dig. Gland trial ! 0006 16 hr .001 .0005 .001 16 hr trial 2 Digestive Gland control 000 trial 16 hr .0007 .0007 trial 2 16 hr .0005 Difference +.001 +.003 -.006 +.008 .000 +.004 +.001 +.001 +003 +.002 +.001 +.004 +.0002 + 0003 +.001 +.001 +.0001 +.0001 +.0002 +0001 +0004 +.0005 .000 +.0002 mo frainme me gea Table 1 continued Enzyme Initial Incubation time Uricase Uric acid control trial 1 8 hr .20 trial 2 8 hr .20 ric acid-kidney trial 1 8 hr .19 trials2 19 8 hr Kidney control trial 0004 8 hr trial 2 o004 8 hr Uric acid control trial 1 8 hr .19 trial 2 8 hr .20 Uric acid-Dig. Gland trial 1 8 hr .19 trial 2 .19 8 hr Dig. Gland control trial 8 hr .0003 trial 2 .0003 8 hr Urease Urea control 8 hr trial 008 trial 2 .007 8 hr Urea-Kidney 8 hr trial .010 trial 8 hr .007 Kidney control trial .008 8 hr trial 2 8 hr .009 Urea control .008 8 hr trial ! trial 2 8 hr .006 Urea- Dig. Gland trial 1 .020 8 hr .017 8 hr trial 2 Dig. Gland control trial! 8 hr .01 trial 2 .009 8 hr Final tion .20 .20 .12 .12 .0005 0004 .19 .20 185 185 0004 0004 .01 .010 .056 .056 .01 .01 .01 .01 .019 .019 .012 .012 Difference 000 000 +.08 +.08 +.0001 +.0001 000 000 +.005 +.005 +.0001 +.0001 +.008 + 012 +.184 +.196 +.008 +.004 +.008 +.016 -.004 +.008 +.008 +.008 nq Urie actd ma a Table 2 All values in mg of substrate converted Production of ammonia from uric acid by uricase Incubation Final NH, Initial NH3 Enzyme time Uric acid control .001 8 hr trial ! .002 8 hr .002 .001 tri,12 Uric acid-kidney 8 hr .022 .004 trial ! 8 hr .005 trial 2 .025 Kidney control .001 .003 8 hr trial .003 trial 2 .001 8 hr Uric acid control 8 hr .001 trial ! .001 8 hr .002 trial 2 .001 Uric acid-digestive gland .010 .005 8 hr trial .008 8 hr .013 trial 2 Digestive Gland control 8 hr .005 .002 trial i .007 .003 8 hr trial 2 mg NH, -.004 +.004 +.072 +.090 +008 +.008 .000 +.004 +020 +.020 +.012 +.016 Bibliography Albrecht (1920). J. Biol. Chem. 45, 395. 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